Stuart Michelson | Researcher Profile | Sotabase

Career

· Chair, Human Systems Division, National Defense Industrial Association - (NDIA)2023–2025

· Chairman, Board Of Directors, Trail Life USA2013–

· Advisory Committee, Reformation Hope2012–2014

· Assoc. Division Chief, Human Centered Engineering Division, Georgia Tech Research Institute2007–

· Organizer, American Venue, International Aerial Robotics Competition (Current)2000–

Publications (31)

Design and synthesis of 8-hydroxy-[1,6]naphthyridines as novel inhibitors of HIV-1 integrase in vitro and in infected cells.

Journal of Medicinal Chemistry · 2003

238

cited

New isomeric classes of topically active ocular hypotensive carbonic anhydrase inhibitors: 5-substituted thieno[2,3-b]thiophene-2-sulfonamides and 5-substituted thieno[3,2-b]thiophene-2-sulfonamides.

Journal of Medicinal Chemistry · 1991

cited

(Acyloxy)alkyl carbamates as novel bioreversible prodrugs for amines: increased permeation through biological membranes.

Journal of Medicinal Chemistry · 1988

cited

Development of orally active oxytocin antagonists: studies on 1-(1-[4-[1-(2-methyl-1-oxidopyridin-3-ylmethyl)piperidin-4-yloxy]-2- methoxybenzoyl]piperidin-4-yl)-1,4-dihydrobenz[d][1,3]oxazin-2-one (L-372,662) and related pyridines.

Journal of Medicinal Chemistry · 1998

cited

Topically active carbonic anhydrase inhibitors. 3. Benzofuran- and indole-2-sulfonamides.

Journal of Medicinal Chemistry · 1990

cited

Identification of MK-944a: a second clinical candidate from the hydroxylaminepentanamide isostere series of HIV protease inhibitors.

Journal of Medicinal Chemistry · 2000

cited

Orally efficacious NR2B-selective NMDA receptor antagonists.

Bioorganic & Medicinal Chemistry Letters · 2003

cited

Inhibitors of glycolic acid oxidase. 4-Substituted 3-hydroxy-1H-pyrrole-2,5-dione derivatives.

Journal of Medicinal Chemistry · 1983

cited

Time- and dose-dependent pharmacokinetics of L-754,394, an HIV protease inhibitor, in rats, dogs and monkeys.

Journal of Pharmacology and Experimental Therapeutics · 1995

cited

Inhibitors of glycolic acid oxidase. 4-substituted 2,4-dioxobutanoic acid derivatives.

Journal of Medicinal Chemistry · 1983

cited

Quantitative structure-activity relationships involving the inhibition of glycolic acid oxidase by derivatives of glycolic and glyoxylic acids.

Journal of Medicinal Chemistry · 1979

cited

Topically active carbonic anhydrase inhibitors. 4. [(Hydroxyalkyl)sulfonyl]benzene and [(hydroxyalkyl)sulfonyl]thiophenesulfonamides.

Journal of Medicinal Chemistry · 1991

cited

Cycloalkylpiperazines as HIV-1 protease inhibitors: enhanced oral absorption

1995

cited

Thieno[2,3-b]furan-2-sulfonamides as topical carbonic anhydrase inhibitors.

Journal of Medicinal Chemistry · 1992

cited

3-substituted thieno[2,3-b][1,4]thiazine-6-sulfonamides. A novel class of topically active carbonic anhydrase inhibitors.

Journal of Medicinal Chemistry · 1994

cited

4-substituted thiophene- and furan-2-sulfonamides as topical carbonic anhydrase inhibitors.

Journal of Medicinal Chemistry · 1992

cited

Nonpeptide oxytocin antagonists: analogs of L-371,257 with improved potency.

Bioorganic & Medicinal Chemistry Letters · 1999

cited

Thiophene derivatives as extremely high affinity P3′ ligands for the hydroxyethylpiperazine class of HIV-1 protease inhibitors

1995

cited

A new hydroxyethylamine class of HIV-1 protease inhibitors with high antiviral potency and oral bioavailability

1994

cited

Substituted alkylpyridines as P3′ ligands for the hydroxyethylpiperazine class of HIV-1 protease inhibitors: Improved pharmacokinetic profiles

1995

cited

Sotabase