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Career

· Distinguished Fellow, NYU Center for Cybersecurity

Publications (52)

Studies on the Synthesis of Nargenicin A1: Highly Stereoselective Synthesis of the Complete Carbon Framework via the Transannular Diels−Alder Reaction of an 18-Membered Macrolide
1996
81
cited
Stereoselective synthesis of (Z,E)-2-bromo-1,3-dienes via the palladium (O) catalyzed cross coupling reactions of 1,1-dibromoolefins and vinylboronic acids
1990
72
cited
Comprehensive survey of combinatorial library synthesis: 2005.
Journal of combinatorial chemistry · 2006
62
cited
Enantioselective synthesis of the bottom half of chlorothricolide. 3. Studies of the steric directing group strategy for stereocontrol in intramolecular Diels-Alder reactions
1991
59
cited
The synthesis and SAR of 2-amino-pyrrolo[2,3-d]pyrimidines: a new class of Aurora-A kinase inhibitors.
Bioorganic & Medicinal Chemistry Letters · 2006
58
cited
Synthetic, x-ray structural and photoluminescence studies on pentamethylcyclopentadienyl derivatives of lanthanum, cerium and praseodymium
1986
55
cited
The formation and crystal and molecular structures of (η5-pentamethylcyclopentadienyl)(η5-cyclopentadienyl)dichloro-titanium, -zirconium and -hafnium
1985
55
cited
The discovery of orally active triaminotriazine aniline amides as inhibitors of p38 MAP kinase.
Journal of Medicinal Chemistry · 2004
45
cited
Novel cytokine release inhibitors. Part I: Triterpenes.
Bioorganic & Medicinal Chemistry Letters · 1998
42
cited
Discovery, SAR, and X-ray structure of novel biaryl-based dipeptidyl peptidase IV inhibitors.
Bioorganic & Medicinal Chemistry Letters · 2006
35
cited
Discovery, SAR and X-ray structure of 1H-benzimidazole-5-carboxylic acid cyclohexyl-methyl-amides as inhibitors of inducible T-cell kinase (Itk).
Bioorganic & Medicinal Chemistry Letters · 2008
29
cited
Synthesis, biological evaluation, and pharmacokinetic study of prolyl-1-piperazinylacetic acid and prolyl-4-piperidinylacetic acid derivatives as VLA-4 antagonists.
Bioorganic & Medicinal Chemistry · 2006
28
cited
Itk kinase inhibitors: initial efforts to improve the metabolical stability and the cell activity of the benzimidazole lead.
Bioorganic & Medicinal Chemistry Letters · 2008
26
cited
Isodicyclopentadienes and related molecules. 44. Analysis of the .pi.-facial preference for complexation of a camphor-derived, enantiomerically pure cyclopentadienyl ligand to CpMCl2 fragments (M = Ti and Zr)
1989
25
cited
Stereoselective formation from a (1S,5S)-(−)-verbenone-derived cyclopentadiene of dimeric and mixed titanium and zirconium dichloride complexes
1989
19
cited
The synthesis and biological evaluation of a novel series of indole PDE4 inhibitors I.
Bioorganic & Medicinal Chemistry Letters · 1998
19
cited
Identified a morpholinyl-4-piperidinylacetic acid derivative as a potent oral active VLA-4 antagonist.
Bioorganic & Medicinal Chemistry Letters · 2005
18
cited
Isodicyclopentadienes and related molecules. 45. (1R)-(-)-Nopol as the source of an optically pure fused cyclopentadienyl ligand. Stereochemical course of complexation to cyclopentadienyltitanium and -zirconium dichloride fragments
1989
18
cited
Orally active indole N-oxide PDE4 inhibitors.
Bioorganic & Medicinal Chemistry Letters · 1998
18
cited
4-[2-[Methyl(2-phenethyl)amino]-2-oxoethyl]-8-(phenylmethoxy)-2- naphthalenecarboxylic acid: a high affinity, competitive, orally active leukotriene B4 receptor antagonist.
Journal of Medicinal Chemistry · 1992
16
cited
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Kevin Moriarty | Researcher Profile | Sotabase | Sotabase